I-Retatrutide (LY3437943)yi-peptide yokwenziwa yesizukulwana esilandelayo eyenziwe njengei-agonist ye-receptor ezintathuijolise kwi-GLP-1, GIP, kunye nee-glucagon receptors. Uyilo lwayo olutsha lweemolekyuli luyahlula kwiiteknoloji zepeptide ze-single- kunye ne-dual-receptor zangaphambili, nto leyo eyenza ukuba ibe yenye yezona zinto zifundwa kakhulu kuphando lwangoku lwe-metabolic.
Ibonelelwa njengomgubo ococekileyo kakhulu,I-RetatrutideInika uzinzo oluhle kakhulu ekuphathweni kwelebhu, ekuthuthweni, nasekugcinweni kwexesha elide. Isetyenziswa kakhulu kuphando lwesayensi olubandakanya i-receptor signaling, ukulawulwa kwe-metabolic, ubunjineli be-peptide, kunye nophando lwe-endocrine.
✔ Ucoceko Oluphezulu (≥98% HPLC)
✔ Umgubo ocoliweyo omhlophe ukuya komhlophe
✔ Uzinzo Oluhle Kakhulu kwiZicelo zoPhando
✔ Ubuchwepheshe be-Agonist ye-Triple Receptor
✔ Ulawulo oluQinisekileyo loMgangatho kunye nokuHlangana kweBatch
✔ Ifanelekile kwi-Advanced Peptide Research
| Into | Inkcazo |
|---|---|
| Igama lemveliso | I-Retatrutide |
| Isithethantonye | LY3437943 |
| Ifomula yeMolekyuli | C221H342N46O68* |
| Ubunzima beMolekyuli | Malunga ne-4731 Da* |
| Inkangeleko | Umgubo oMhlophe oPhilisiweyo |
| Ubunyulu | ≥98% nge-HPLC |
| Indawo yokugcina izinto | -20°C Kucetyiswa |
| Ukunyibilika | Amanzi Anyibilikayo |
| Isicelo | Uphando lweLebhu Kuphela |
*Iinkcukacha zinokwahluka ngokweqela lokwenziwa kunye nemigangatho yohlalutyo.
| Igama lemveliso | Inombolo ye-CAS |
|---|---|
| I-AOD-9604 | 221231-10-3 |
| I-BPC-157 | 137525-51-0 |
| I-PT-141 / i-Bremelanotide Acetate | 189691-06-3 |
| I-CJC-1295 | 863288-34-0 |
| I-GHK-Cu | 89030-95-5 |
| I-GHRP-2 | 158861-67-7 |
| I-Hexarelin | 140703-51-1 |
| IGF-1 LR3 | 946870-92-4 |
| Ipamorelin | 170851-70-4 |
| I-KPV / Alpha MSH (11-13) | 67727-97-3 |
| I-L-Arginine | 74-79-3 |
| I-MOTS-C | 1627580-64-6 |
| I-Oxytocin | 50-56-6 |
| I-PDA | 106-50-3 |
| Selank | 129954-34-3 |
| I-Semax | 80714-61-0 |
| ISermorelin | 86168-78-7 |
| I-SS-31 (Lyo) / I-Elamipretide | 736992-21-5 |
| Isiqwenga seTB500 | 476014-70-7 |
| I-Tesamorelin | 218949-48-5 |
| I-Thymogen / i-Oglufanide | 38101-59-6 |
| Thymosin Alpha-1 / Thymalfasin | 62304-98-7 |
| I-Thymosin Beta-4 | 77591-33-4 |
| TB500 | 885340-08-9 |
| I-NVG-291 | 2135482-62-7 |
| CB4211 | 2361287-87-0 |
| I-DSIP | 62568-57-4 |
| I-Epitalon | 307297-39-8 |
| IGonadorelin | 33515-09-2 |
| LL-37 | 154947-19-0 |
| I-Melanotan II | 121062-08-6 |
| MK-0616 | 2249825-14-7 |
| I-NAD+ | 53-84-9 |
| I-Pamorelin | 57773-63-1 |
| I-PTD-DBM | 1241682-11-0 |
| Isiqwenga 176-191 | 66004-57-7 |
| I-VIP | 40077-57-4 |
| PE-22-28 | 1136689-11-0 |
I-Retatrutide yenzelwe ukusebenza ngaxeshanye ukuze isebenze ii-receptors ezintathu ze-metabolic hormone ngaxeshanye:
Oku kunxulumene nokulawula inkanuko, iindlela zokukhupha isisu, kunye neendlela zokubonisana ezinxulumene neswekile.
Ibandakanyeka ekuqondeni izondlo, ukuhanjiswa kwe-insulin, kunye neenkqubo zokulawula imetabolism.
Inxulunyaniswa nenkcitho yamandla, imetabolism yamafutha, kunye neendlela zokulungelelanisa imetabolism.
Ukusebenza okudibeneyo kwezi nkqubo zintathu zee-receptor kwenza iRetatrutide ibe yinxalenye yophando eyahlukileyo yokuphanda ukusebenzisana okuntsonkothileyo kwe-metabolic kunye neempendulo zebhayoloji ezisebenzisa iindlela ezininzi.
I-Retatrutide ibe yinto ebalulekileyo kwiindawo ezahlukeneyo zophando lwesayensi, kuquka:
Abaphandi bayaqhubeka nokuphonononga iprofayili yayo eyahlukileyo ye-triple-agonist kunye neziphumo zayo ezinokubakho kuphuhliso lwe-peptide kwixesha elizayo.
Yonke ibhetshi yeRetatrutide kufuneka ivavanywe ngokucokisekileyo, kuquka:
ISatifikethi soHlalutyo (i-COA) singanikezelwa xa siceliwe ukuqinisekisa umgangatho wemveliso kunye nokulandeleka kwayo.
Ukugcina uzinzo olufanelekileyo lwe-peptide:
Ugcino Lwexesha Elide
Emva koHlaziyo loMgaqo-siseko
Iimeko ezifanelekileyo zokugcina izinto zinceda ukugcina ukuthembeka kwe-peptide kunye nokusebenza kohlalutyo.
Iindlela zokupakisha ezikhoyo zingabandakanya:
Ubungakanani obukhulu kunye neenkonzo zokupakisha ze-OEM ziyafumaneka kwimibutho yophando efanelekileyo.
I-Retatrutide inikezelwa kuphela kuphando lwelabhoratri kunye neenjongo zohlalutyo. Le mveliso ayivumelekanga ukusetyenziswa ngabantu, ukusetyenziswa kwezonyango, ukusetyenziswa kwezonyango, okanye iinkqubo zokuxilonga. Abaphandi banoxanduva lokuqinisekisa ukuthotyelwa kwayo yonke imigaqo efanelekileyo kunye nezikhokelo zeziko.